SCHEMBL5199805

SCHEMBL5199805

CC(C)(C)OC(=O)ON1CCC[C@H]1CNc1ccc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 16/20 0.51
CHRM1 P11229 4/20 0.50
HTR2A P28223 3/20 0.50
CYP2D6 P10635 1/20 0.44
ACACB O00763 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13708522 0.87 MCHR1 (0.52) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4485852 0.82 MCHR1 (0.59) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL4488028 0.82 MCHR1 (0.59) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL2328512 0.75 MCHR1 (0.66) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2325038 0.73 MCHR1 (0.53) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4511689 0.70 MCHR1 (0.68) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4493104 0.70 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL13920424 0.69 MCHR1 (0.64) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2323028 0.68 MCHR1 (1.00) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2326750 0.68 MCHR1 (0.67) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737823-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2007-01-03 EP disclosed
WO-2005103002-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed