SCHEMBL5201514

SCHEMBL5201514

NCC(N)c1ccc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 14/20 0.52
CHRM1 P11229 3/20 0.51
HTR2A P28223 3/20 0.51
CYP2D6 P10635 1/20 0.51
AKT2 P31751 3/20 0.41
ACACB O00763 2/20 0.39
ADK P55263 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4475875 0.85 MCHR1 (0.49) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL2324515 0.79 MCHR1 (0.56) MCHR1CHRM1HTR2ACYP2D6ADK
SCHEMBL5228441 0.78 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL5226134 0.78 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL6366478 0.77 MCHR1 (0.57) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL4481796 0.76 MCHR1 (0.56) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4475382 0.76 MCHR1 (0.56) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4481552 0.76 MCHR1 (0.69) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL6366023 0.76 MCHR1 (0.56) MCHR1CHRM1HTR2ACYP2D6ACACB
SCHEMBL5198730 0.75 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737823-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2007-01-03 EP disclosed
WO-2005103002-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed