SCHEMBL5201869

SCHEMBL5201869

Cc1ncc(-c2ccncn2)n1C(C)C.O=C(Cl)CCl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 18/20 0.45
KCNH2 Q12809 7/20 0.45
CDK1 P06493 4/20 0.40
CDK4 P11802 4/20 0.40
CCNT1 O60563 1/20 0.40
CCNB1 P14635 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CCNA2 P20248 1/20 0.40
CCND1 P24385 1/20 0.40
CCNE1 P24864 1/20 0.40
CCND3 P30281 1/20 0.40
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
CSNK1A1 P48729 1/20 0.40
CSNK1D P48730 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CDK7 P50613 1/20 0.40
CDK9 P50750 1/20 0.40
CCNH P51946 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4505142 0.87 CDK2 (0.49) CDK2KCNH2CDK1CDK4CCNT1
Acetic Acid SCHEMBL4253108 0.68 CDK2 (0.57) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL3207123 0.68 CDK2 (0.60) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL3217346 0.68 CDK2 (0.57) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL4253102 0.67 CDK2 (0.53) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL278830 0.65 CDK2 (0.56) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL4508243 0.62 CDK2 (1.00) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL8950388 0.62 PIK3CA (0.41) MAPK9CSNK1A1GSK3B
SCHEMBL1447341 0.61 CDK2 (0.81) CDK2KCNH2CDK1CDK4CCNT1
SCHEMBL22322804 0.60 CYP2D6 (0.40) GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748999-A1 IMIDAZOLO-5-YL-2-ANILINOPYRIMIDINES AS AGENTS FOR THE INHIBITION OF CELL PROLIFERATION AstraZeneca AB (SE) 2007-02-07 EP disclosed
WO-2005075461-A1 IMIDAZOLO-5-YL-2-ANILINOPYRIMIDINES AS AGENTS FOR THE INHIBITION OF CELL PROLIFERATION ASTRAZENECA AB (SE) 2005-08-18 WO disclosed