SCHEMBL5209380

SCHEMBL5209380

Cc1ccc(-c2cc3cc(C(=O)O)ccc3o2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.58
TP53 P04637 1/20 0.55
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 2/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
HPGD P15428 1/20 0.49
ESR1 P03372 1/20 0.49
ESR2 Q92731 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
CSNK2A2 P19784 1/20 0.47
CSNK2B P67870 1/20 0.47
CSNK2A1 P68400 1/20 0.47
TNKS O95271 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5210930 0.88 HDAC6 (0.56) MAOBALDH1A1KDM4EGAAMAPT
SCHEMBL3922682 0.86 ESR1 (0.68) MAOBTP53ALDH1A1KDM4EMAPT
SCHEMBL977340 0.86 FFAR1 (0.58) MAOBESR1ESR2TNKSHDAC6
SCHEMBL3121270 0.85 NPC1 (0.52) ALDH1A1KDM4EMAPTESR1ESR2
SCHEMBL978657 0.84 APP (0.58) MAOBTP53ALDH1A1KDM4EGAA
SCHEMBL11855280 0.84 MAOB (0.57) MAOBTP53ALDH1A1KDM4EGAA
SCHEMBL11855285 0.84 MAOB (0.57) MAOBTP53ALDH1A1KDM4EGAA
SCHEMBL11826060 0.82 HDAC6 (0.52) MAOBALDH1A1KDM4EGAAMAPT
SCHEMBL3377936 0.81 FFAR1 (0.64) MAOBESR1ESR2TNKSP2RY14
SCHEMBL27521215 0.81 FFAR1 (0.51) MAOBTP53ESR1ESR2TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed
EP-1039899-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
EP-1040103-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-10-04 EP disclosed
WO-1999032100-A2 PHARMACEUTICAL COMPOSITION FOR ANTAGONIZING CCR5 COMPRISING ANILIDE DERIVATIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed
WO-1999032468-A1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-01 WO disclosed