SCHEMBL5215892

SCHEMBL5215892

CC(C)CNC(=O)c1cnc(Nc2ccc(Cl)c(Cl)c2)cc1C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 14/20 0.55
HPGD P15428 1/20 0.46
IRAK4 Q9NWZ3 4/20 0.45
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5213789 0.87 CNR2 (0.73) CNR2CYP1A2
SCHEMBL5213486 0.86 CNR2 (0.58) CNR2IRAK4NPSR1L3MBTL1
SCHEMBL5213870 0.85 CNR2 (0.56) CNR2IRAK4
SCHEMBL4650388 0.84 CNR2 (0.76) CNR2HPGDIRAK4CYP1A2
SCHEMBL5216312 0.84 CNR2 (0.65) CNR2IRAK4
SCHEMBL5212556 0.83 CNR2 (0.70) CNR2CYP1A2
SCHEMBL5213108 0.83 CNR2 (0.69) CNR2IRAK4NPSR1CYP1A2
SCHEMBL5212199 0.83 CNR2 (0.70) CNR2IRAK4CYP1A2
SCHEMBL5787298 0.82 CNR2 (0.72) CNR2CYP1A2
SCHEMBL5212174 0.81 CNR2 (0.74) CNR2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565442-B1 PYRIDINE DERIVATIVES AS CB2 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2007-11-14 EP claimed
EP-1565442-B1 PYRIDINE DERIVATIVES AS CB2 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2007-11-14 EP disclosed
US-20060240048-A1 Pyridine derivatives as cb2 receptor modulators GLAXO GROUP LIMITED (GB) 2006-10-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060240048-A1 Pyridine derivatives as cb2 receptor modulators CNR2, CNR1, TRPV1 CNR2 1/4885HPGD 524/4885IRAK4 1243/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.