SCHEMBL5219571

SCHEMBL5219571

O=C(O)NC1CCN(c2ccc3ccccc3n2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.55
KDM4E B2RXH2 7/20 0.54
ALDH1A1 P00352 6/20 0.54
CYP3A4 P08684 2/20 0.54
HSD17B10 Q99714 2/20 0.54
HTR3E A5X5Y0 2/20 0.51
HTR3B O95264 2/20 0.51
CYP1A2 P05177 2/20 0.51
HTR3A P46098 2/20 0.51
HTR3D Q70Z44 2/20 0.51
HTR3C Q8WXA8 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
USP2 O75604 1/20 0.51
ADRB1 P08588 1/20 0.51
HTR1A P08908 1/20 0.51
HTR2C P28335 1/20 0.51
MAPK1 P28482 1/20 0.51
SLC6A4 P31645 1/20 0.51
HTR7 P34969 1/20 0.51
HTT P42858 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2630866 0.86 PDE10A (0.53) HRH3KDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL27649158 0.84 PDE10A (0.69) HRH3KDM4EALDH1A1HSD17B10HTR3E
SCHEMBL28803641 0.82 HRH3 (0.58) HRH3KDM4EALDH1A1CYP3A4HSD17B10
Hydrochloric Acid SCHEMBL16648730 0.81 HRH3 (0.57) HRH3KDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL2596336 0.80 PDE10A (0.81) PDE10A
SCHEMBL1727542 0.79 HRH3 (0.52) HRH3KDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL3289098 0.78 DRD3 (0.43) KDM4EALDH1A1CYP3A4HSD17B10PDE10A
SCHEMBL2631079 0.78 HRH3 (0.65) HRH3KDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL31381307 0.78 PDE10A (0.68) HRH3KDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL16769735 0.78 HRH3 (0.57) HRH3KDM4EALDH1A1CYP3A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664025-B1 PYRROL DERIVATIVES WITH ANTIBACTERIAL ACTIVITY ASTRAZENECA AB (SE) 2007-09-19 EP disclosed