SCHEMBL5220697

SCHEMBL5220697

CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@H](O)CNC(C)Cc2cccc(Cl)c2)cc(N2CCCCS2(O)O)c1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.65
BACE2 Q9Y5Z0 19/20 0.65
CTSD P07339 18/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224785 1.00 BACE1 (0.65) BACE1BACE2CTSD
Hydrochloric Acid SCHEMBL5222028 0.99 BACE1 (0.66) BACE1BACE2CTSD
Hydrochloric Acid SCHEMBL5222023 0.99 BACE1 (0.66) BACE1BACE2CTSD
SCHEMBL5220703 0.94 BACE1 (0.74) BACE1BACE2CTSD
Hydrochloric Acid SCHEMBL5222013 0.93 BACE1 (0.76) BACE1BACE2CTSD
SCHEMBL5218924 0.91 BACE1 (0.64) BACE1BACE2CTSD
SCHEMBL5219269 0.91 BACE1 (0.64) BACE1BACE2CTSD
SCHEMBL5226901 0.91 BACE1 (0.71) BACE1BACE2CTSD
SCHEMBL5226905 0.91 BACE1 (0.71) BACE1BACE2CTSD
Hydrochloric Acid SCHEMBL5221425 0.91 BACE1 (0.63) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP claimed