SCHEMBL5221200

SCHEMBL5221200

CCc1c(-c2ccc(O)cc2)nn(-c2cc(Cl)cc(Cl)c2)c1-c1ccc(O)cc1.CCc1c(-c2ccc(O)cc2)nn(-c2ccc(Cl)cc2C)c1-c1ccc(O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
GMNN O75496 1/20 0.49
USP2 O75604 1/20 0.49
LMNA P02545 1/20 0.49
ESR1 P03372 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
ALOX12 P18054 1/20 0.49
NFKB1 P19838 1/20 0.49
MAPK1 P28482 1/20 0.49
CYP2C19 P33261 1/20 0.49
THPO P40225 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5222191 0.94 CNR2 (0.49) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5215497 0.89 ESR1 (0.60) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5219512 0.83 CNR2 (0.61) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5214017 0.82 MAPK1 (0.51) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5218508 0.82 CNR1 (0.46) CNR2CNR1PPARA
SCHEMBL5215832 0.81 ESR1 (0.56) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5221678 0.81 ESR1 (0.69) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5214152 0.80 ESR1 (0.42) KDM4EGMNNUSP2LMNAESR1
SCHEMBL5218760 0.78 CNR1 (0.43) CNR2CNR1PPARA
SCHEMBL5220810 0.77 MAPT (0.53) KDM4EGMNNUSP2LMNAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102753-B1 PYRAZOLES AS ESTROGEN RECEPTOR MODULATORS NOVARTIS VACCINES & DIAGNOSTIC (US) 2007-02-28 EP disclosed