SCHEMBL5221950

SCHEMBL5221950

COc1cc2nccc(Oc3c(C)cccc3F)c2cc1OC

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.55
PDGFRA P16234 4/20 0.54
PDGFRB P09619 1/20 0.54
KDR P35968 3/20 0.53
AXL P30530 1/20 0.53
SRC P12931 1/20 0.52
TGFBR1 P36897 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3892996 0.83 PDGFRA (0.53) EGFRPDGFRAPDGFRBKDR
SCHEMBL13739661 0.81 SRC (0.60) EGFRPDGFRAPDGFRBKDRSRC
SCHEMBL3906011 0.79 KDR (0.54) PDGFRAKDRSRCTGFBR1
SCHEMBL3895896 0.79 PDGFRA (0.49) EGFRPDGFRAPDGFRBKDR
SCHEMBL14967538 0.79 PDGFRB (0.57) EGFRPDGFRAPDGFRBKDRAXL
SCHEMBL3927341 0.79 FGFR2 (0.58) EGFRPDGFRAPDGFRBKDR
SCHEMBL25826950 0.79 EGFR (0.60) EGFRPDGFRAPDGFRB
SCHEMBL5824622 0.78 AXL (0.52) EGFRPDGFRAKDRAXLSRC
SCHEMBL7485861 0.78 EGFR (0.66) EGFRPDGFRAPDGFRBSRCTGFBR1
SCHEMBL14966472 0.77 PDGFRB (0.58) EGFRPDGFRAPDGFRBKDRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1827434-A2 QUINOLINES AND QUINAZOLINE ANALOGS AND THEIR USE AS MEDICAMENTS FOR TREATING CANCER Amgen Inc. (US) 2007-09-05 EP disclosed
WO-2006060318-A2 QUINOLINES AND QUINAZOLINE ANALOGS AND THEIR USE AS MEDICAMENTS FOR TREATING CANCER AMGEN INC. (US) 2006-06-08 WO disclosed