SCHEMBL5223219

SCHEMBL5223219

COc1ccc(N(C(=O)O)c2nc3cc(N(C)c4ccnc(Nc5ccc(CS(C)(=O)=O)cc5)n4)ccc3n2C)c(C(C)(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.47
AURKA O14965 1/20 0.44
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226472 0.94 KDR (0.44) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL5227304 0.94 KDR (0.52) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5226925 0.90 KDR (0.44) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL5227350 0.90 KDR (0.52) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL4981188 0.86 KDR (0.49) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL5227882 0.84 KDR (0.49) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL5225387 0.83 KDR (0.57) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL5226596 0.81 KDR (0.52) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL14263363 0.81 KDR (0.53) KDRAURKACYP3A4CYP2D6CYP2C9
SCHEMBL6407659 0.81 KDR (0.54) KDRAURKACYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP claimed