SCHEMBL5226400

SCHEMBL5226400

COC(=O)C(CCSc1cccc(-c2cccc(-c3cccc4c3oc3ccccc34)c2)c1)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.42
GGPS1 O95749 1/20 0.39
KLK5 Q9Y337 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
NPC1 O15118 1/20 0.38
PLIN1 O60240 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
PLIN5 Q00G26 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ABHD5 Q8WTS1 1/20 0.38
ALOX5 P09917 1/20 0.37
CTSS P25774 2/20 0.37
CTSK P43235 2/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
GSTP1 P09211 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3873193 0.94 EPHX2 (0.42) EPHX2GGPS1KLK5KDM4EALDH1A1
SCHEMBL13897379 0.92 GSTP1 (0.42) EPHX2GGPS1KLK5KDM4EALDH1A1
SCHEMBL3862993 0.92 FNTA (0.44) EPHX2GGPS1ALDH1A1ALOX5CTSS
SCHEMBL3871194 0.92 GSTP1 (0.42) EPHX2GGPS1KLK5KDM4EALDH1A1
SCHEMBL13897413 0.90 EPHX2 (0.44) EPHX2GGPS1KLK5KDM4EALDH1A1
SCHEMBL3864792 0.87 FNTA (0.43) EPHX2GGPS1KDM4EALDH1A1NPC1
SCHEMBL3863222 0.86 PPARA (0.43) EPHX2GGPS1ALOX5CTSSCTSK
SCHEMBL13897480 0.86 PPARA (0.43) EPHX2GGPS1ALOX5CTSSCTSK
SCHEMBL3867006 0.86 BCHE (0.44) EPHX2GGPS1KLK5KDM4EALDH1A1
SCHEMBL3863211 0.85 GGPS1 (0.45) EPHX2GGPS1KLK5MAPTALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1814869-A2 SUBSTITUTED AMINO ACIDS AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS The Institutes for Pharmaceutical Discovery, LLC (US) 2007-08-08 EP claimed
WO-2006055725-A2 SUBSTITUTED AMINO ACIDS AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2006-05-26 WO claimed