SCHEMBL5226590

SCHEMBL5226590

Cn1c(N(C(=O)O)c2ccc(F)cc2)nc2cc(Nc3ccnc(Cl)n3)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
USP2 O75604 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
AURKA O14965 1/20 0.38
BRAF P15056 3/20 0.36
NPC1 O15118 5/20 0.36
RAB9A P51151 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228478 0.92 NPC1 (0.41) TP53BRAFNPC1RAB9AMAPT
SCHEMBL5230055 0.89 BRAF (0.39) MEN1KMT2ALMNAMAPK1ALDH1A1
SCHEMBL5226236 0.89 BRAF (0.45) BRAFNPC1RAB9AMAPTHDAC6
SCHEMBL4978728 0.88 BRAF (0.37) GRM5MEN1KMT2AUSP2CYP1A2
SCHEMBL5224254 0.82 KDR (0.38) GRM5CYP3A4CYP2C19CYP2D6CYP2C9
SCHEMBL4980380 0.80 BRAF (0.37) AURKABRAFNPC1RAB9AMAPT
SCHEMBL5225363 0.80 RAF1 (0.39) AURKABRAFNPC1RAB9AMAPT
SCHEMBL4983383 0.80 NPC1 (0.38) BRAFNPC1RAB9AMAPTPOLB
SCHEMBL4983374 0.79 BRAF (0.44) CYP3A4BRAFNPC1RAB9A
SCHEMBL4980603 0.78 BRAF (0.39) MEN1KMT2ALMNAMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed