SCHEMBL5226887

SCHEMBL5226887

OC(COc1ccc2sc(-c3ccccc3)nc2c1)CN1C[CH]N(c2ccc3[nH]ncc3c2)CC1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.50
PRMT5 O14744 2/20 0.48
WDR77 Q9BQA1 2/20 0.48
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205691 0.86 KCNH2 (0.51) KCNH2PRMT5WDR77CYP1A2CYP3A4
SCHEMBL7005719 0.81 CYP3A4 (0.52) CYP1A2CYP3A4CYP2C9
SCHEMBL4864558 0.80 CYP3A4 (0.67) CYP1A2CYP3A4CYP2C9
SCHEMBL4033617 0.77 CYP3A4 (0.55) CYP1A2CYP3A4CYP2C9
SCHEMBL6207329 0.77 KCNH2 (0.49) KCNH2PRMT5WDR77CYP1A2CYP3A4
SCHEMBL5228562 0.77 CYP3A4 (0.48) CYP1A2CYP3A4CYP2C9
SCHEMBL5223317 0.73 KCNH2 (0.47) KCNH2PRMT5WDR77CYP3A4
SCHEMBL5228642 0.73 CYP1A2 (0.47) CYP1A2CYP3A4CYP2C9
SCHEMBL5965111 0.73 CYP3A4 (0.53) CYP1A2CYP3A4CYP2C9
SCHEMBL5901541 0.73 CYP3A4 (0.53) CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806346-A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors CV THERAPEUTICS, INC. (US) 2007-07-11 EP disclosed
EP-1567525-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2005-08-31 EP disclosed
WO-2004052887-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2004-06-24 WO disclosed