SCHEMBL5227045

SCHEMBL5227045

CN(c1ccc2c(c1)nc(NCc1ccc(Cl)cc1)n2C)c1ccnc(Nc2cccc(CS(=O)(=O)O)c2)n1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDR P35968 20/20 0.56
CYP3A4 P08684 4/20 0.56
CYP2D6 P10635 4/20 0.56
CYP2C9 P11712 4/20 0.56
CYP2C19 P33261 4/20 0.56
KIT P10721 2/20 0.52
PDGFRA P16234 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5229088 0.99 KDR (0.55) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4980819 0.90 KDR (0.71) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4980945 0.89 KDR (0.70) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4980459 0.88 KDR (0.62) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4976821 0.88 KDR (0.53) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14263351 0.88 KDR (0.58) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4977042 0.88 KDR (0.53) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14263452 0.88 KDR (0.52) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4976772 0.88 KDR (0.62) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4980109 0.88 KDR (0.52) KDRCYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP claimed