SCHEMBL5227437

SCHEMBL5227437

CC(C)c1cccc(CNCC(O)C2Cc3cccc(c3)OCCCCCC(=O)N(C)C(C)C(=O)N2)c1

nearest known ligand 0.69

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.69
CTSD P07339 8/20 0.69
CTSE P14091 4/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2352364 1.00 BACE1 (0.69) BACE1CTSDCTSE
SCHEMBL2355050 1.00 BACE1 (0.69) BACE1CTSDCTSE
SCHEMBL2354066 1.00 BACE1 (0.69) BACE1CTSDCTSE
SCHEMBL2353525 0.99 BACE1 (0.68) BACE1CTSDCTSE
SCHEMBL2351551 0.98 BACE1 (0.68) BACE1CTSDCTSE
SCHEMBL2349597 0.91 BACE1 (0.63) BACE1CTSDCTSE
SCHEMBL2351687 0.90 BACE1 (0.76) BACE1CTSDCTSE
SCHEMBL2354054 0.90 BACE1 (0.76) BACE1CTSDCTSE
SCHEMBL2349979 0.83 BACE1 (0.73) BACE1CTSDCTSE
SCHEMBL2353194 0.82 BACE1 (0.43) BACE1CTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838680-A2 MACROCYCLIC COMPOUNDS AND COMPOSITIONS USEFUL AS BACE INHIBITORS Novartis AG (CH) 2007-10-03 EP disclosed
WO-2006074940-A2 MACROCYCLIC COMPOUNDS AND COMPOSITIONS USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2006-07-20 WO disclosed