SCHEMBL5227870

SCHEMBL5227870

Cc1ccc(NC(=O)CN2CCN(CC(O)COc3ccc4sc(C)nc4c3)CC2)c(Cl)c1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.72
CYP1A2 P05177 2/20 0.69
CYP2C9 P11712 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6284854 0.88 CYP3A4 (0.86) CYP3A4CYP1A2CYP2C9
SCHEMBL6285300 0.88 CYP3A4 (0.86) CYP3A4CYP1A2CYP2C9
SCHEMBL5225565 0.87 CYP3A4 (0.76) CYP3A4CYP1A2CYP2C9
SCHEMBL4033917 0.86 CYP3A4 (0.84) CYP3A4CYP1A2CYP2C9
SCHEMBL5226211 0.84 CYP3A4 (0.91) CYP3A4CYP1A2CYP2C9
SCHEMBL4863319 0.84 CYP3A4 (0.77) CYP3A4CYP1A2CYP2C9
SCHEMBL6285110 0.84 CYP3A4 (0.79) CYP3A4CYP1A2CYP2C9
SCHEMBL6280182 0.84 CYP3A4 (0.79) CYP3A4CYP1A2CYP2C9
SCHEMBL6285120 0.84 CYP3A4 (1.00) CYP3A4CYP1A2CYP2C9
SCHEMBL5227719 0.84 CYP3A4 (0.83) CYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339701-B1 HETEROARYL ALKYL PIPERAZINE DERIVATIVES AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS INC (US) 2007-02-14 EP claimed
EP-1339701-B1 HETEROARYL ALKYL PIPERAZINE DERIVATIVES AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS INC (US) 2007-02-14 EP disclosed