SCHEMBL5229414

SCHEMBL5229414

O=C(O)c1n[nH]c2c1CCc1[nH]ncc1-2

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 13/20 0.49
CDK2 P24941 13/20 0.49
CCNA1 P78396 13/20 0.49
HCAR2 Q8TDS4 5/20 0.45
KMT2A Q03164 1/20 0.45
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229284 0.87 CCNA2 (0.58) CCNA2CDK2CCNA1
SCHEMBL5230280 0.80 CCNA2 (0.57) CCNA2CDK2CCNA1KMT2A
SCHEMBL3206132 0.73 GSR (0.53) CDK2HCAR2KMT2ATSHR
SCHEMBL28577870 0.72 NPC1 (0.42) HCAR2KMT2ATSHR
SCHEMBL5233166 0.72 CCNA2 (0.78) CCNA2CDK2CCNA1
Hydrochloric Acid SCHEMBL6792455 0.72 CCNA2 (0.74) CCNA2CDK2CCNA1KMT2A
SCHEMBL5231909 0.70 HCAR2 (0.49) HCAR2KMT2ATSHR
SCHEMBL3517436 0.70 HCAR2 (0.43) HCAR2KMT2ATSHR
SCHEMBL5227895 0.69 CCNA2 (0.82) CCNA2CDK2CCNA1
SCHEMBL6799888 0.68 CCNA2 (0.80) CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478357-B1 TRICYCLIC PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS PFIZER ITALIA SRL (IT) 2007-01-31 EP claimed
CN-109384793-B Thiol compound with HDAC6 inhibitory activity and application thereof 沈阳药科大学 2021-05-07 CN disclosed