SCHEMBL5230128

SCHEMBL5230128

Cc1n[nH]c(CN2CCN(C(=O)O)C(C)C2)c1Oc1cc(Cl)cc(C#N)c1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.46
CYP3A4 P08684 2/20 0.40
CCR1 P32246 1/20 0.38
CHRM4 P08173 2/20 0.36
PTGDR2 Q9Y5Y4 8/20 0.36
MGLL Q99685 2/20 0.33
EGLN1 Q9GZT9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226802 0.86 KCNH2 (0.50) KCNH2CYP3A4MGLL
SCHEMBL509996 0.82 KCNH2 (0.50) KCNH2CYP3A4
SCHEMBL508346 0.81 KCNH2 (0.54) KCNH2CYP3A4
SCHEMBL509154 0.81 KCNH2 (0.48) KCNH2CYP3A4MGLL
SCHEMBL1347408 0.80 KCNH2 (0.48) KCNH2CYP3A4
SCHEMBL14540417 0.79 KCNH2 (0.47) KCNH2CYP3A4MGLL
SCHEMBL509896 0.79 KCNH2 (0.50) KCNH2CYP3A4
SCHEMBL10250900 0.74 KCNH2 (0.78) KCNH2CYP3A4
SCHEMBL509378 0.73 KCNH2 (0.62) KCNH2CYP3A4
SCHEMBL14302751 0.72 KCNH2 (0.64) KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377556-B1 PYRAZOLE DERIVATIVES FOR TREATING HIV PFIZER LTD (GB) 2007-04-04 EP claimed