SCHEMBL5235146

SCHEMBL5235146

O=C1CCCN1/N=C(\Cc1ccnc2ccccc12)c1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.36
MAPT P10636 2/20 0.35
RECQL P46063 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
THRB P10828 1/20 0.35
TGFBR1 P36897 1/20 0.35
MAPK14 Q16539 1/20 0.35
LMNA P02545 3/20 0.35
DRD4 P21917 2/20 0.35
ALDH1A1 P00352 2/20 0.34
RAB9A P51151 2/20 0.34
KDM4E B2RXH2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
FAAH O00519 1/20 0.34
LOXL2 Q9Y4K0 1/20 0.34
FAP Q12884 1/20 0.34
BCHE P06276 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5235150 1.00 CYP1A2 (0.40) CYP1A2GAAMAPTRECQLMEN1
SCHEMBL5240230 0.91 CYP1A2 (0.45) CYP1A2GAAMAPTMEN1KMT2A
SCHEMBL5240236 0.91 CYP1A2 (0.45) CYP1A2GAAMAPTMEN1KMT2A
SCHEMBL5239591 0.89 AR (0.39) CYP1A2GAAMEN1KMT2ALMNA
SCHEMBL5233927 0.89 KDR (0.38) CYP1A2LMNAALDH1A1KDM4ESMN1; SMN2
SCHEMBL5233924 0.89 KDR (0.38) CYP1A2LMNAALDH1A1KDM4ESMN1; SMN2
SCHEMBL5239587 0.89 AR (0.39) CYP1A2GAAMEN1KMT2ALMNA
SCHEMBL5238769 0.85 CYP1A2 (0.40) CYP1A2MAPTLMNAALDH1A1RAB9A
SCHEMBL5238764 0.85 CYP1A2 (0.40) CYP1A2MAPTLMNAALDH1A1RAB9A
SCHEMBL5238619 0.85 KDR (0.35) CYP1A2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed