SCHEMBL5240701

SCHEMBL5240701

CC(Br)CCOCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP2C19 P33261 1/20 0.41
NAAA Q02083 1/20 0.41
CA1 P00915 4/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
VCP P55072 1/20 0.40
TACR1 P25103 2/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL155702 0.84 TSHR (0.56) TSHRTDP1L3MBTL1CYP2C19NAAA
SCHEMBL14763820 0.84 TSHR (0.56) TSHRTDP1L3MBTL1CYP2C19NAAA
SCHEMBL9841232 0.83 TSHR (0.50) TSHRTDP1L3MBTL1CYP2C19NAAA
SCHEMBL10911338 0.83 TSHR (0.50) TSHRTDP1L3MBTL1CYP2C19NAAA
SCHEMBL9841231 0.83 TSHR (0.50) TSHRTDP1L3MBTL1CYP2C19NAAA
SCHEMBL31193586 0.81 TSHR (0.44) TSHRTDP1L3MBTL1CA1CA2
SCHEMBL4781157 0.81 TSHR (0.52) TSHRTDP1L3MBTL1CYP2C19CA1
SCHEMBL2873754 0.81 TSHR (0.52) TSHRTDP1L3MBTL1CYP2C19NAAA
SCHEMBL20582042 0.81 TSHR (0.52) TSHRTDP1L3MBTL1CYP2C19CA1
SCHEMBL14193191 0.81 TSHR (0.52) TSHRTDP1L3MBTL1CYP2C19TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189505-A Tricyclic gyrase inhibitors as antibacterial agents TRIUS THERAPEUTICS INC 2015-12-23 CN disclosed
CN-1968954-A Thienopyridine Derivatives SANKYO CO (JP) 2007-05-23 CN disclosed
EP-1764367-A1 THIENOPYRIDINE DERIVATIVES Sankyo Company, Limited (JP) 2007-03-21 EP disclosed