SCHEMBL5243113

SCHEMBL5243113

CCOc1cc(-c2ccnn2-c2ccc(OC)cc2)ccc1OC(F)F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 1/20 0.46
PDE4D Q08499 8/20 0.44
MAPT P10636 3/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PDE4B Q07343 1/20 0.39
USP2 O75604 1/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GLA P06280 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
DGAT1 O75907 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3606259 0.91 NR3C2 (0.48) NR3C2PDE4DMAPTLMNAHPGD
SCHEMBL3611670 0.90 NR3C2 (0.47) NR3C2PDE4DMAPTLMNAALDH1A1
SCHEMBL3614491 0.83 MAPK9 (0.43) NR3C2PDE4DMAPTLMNAALDH1A1
SCHEMBL3612122 0.81 NR3C2 (0.47) NR3C2MAPTKDM4EALDH1A1HPGD
SCHEMBL3609867 0.79 NR3C2 (0.57) NR3C2PDE4DMAPTLMNAALDH1A1
SCHEMBL3609486 0.76 NR3C2 (0.51) NR3C2MAPTKDM4ELMNAALDH1A1
SCHEMBL3594420 0.73 NR3C2 (0.51) NR3C2MAPTKDM4ELMNAALDH1A1
SCHEMBL13343000 0.72 PDE4A (0.47) PDE4DPDE4B
SCHEMBL3608828 0.72 PDE4A (0.47) PDE4DPDE4B
SCHEMBL15556699 0.71 NR3C2 (0.54) NR3C2MAPTKDM4ELMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799673-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceuticals Corporation (US) 2007-06-27 EP disclosed
WO-2006044528-A1 PYRAZOLE DERIVATIVES AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2006-04-27 WO disclosed