SCHEMBL5243758

SCHEMBL5243758

Cc1cncc(-c2nnc(SCCCN3C[C@@H]4C[C@@]4(c4ccc(Br)cc4)C3)n2C)c1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 20/20 0.67
DRD3 P35462 19/20 0.67
DRD2 P14416 15/20 0.67
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11914551 1.00 KCNH2 (0.67) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL5244397 1.00 KCNH2 (0.67) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL378506 1.00 KCNH2 (0.67) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL5244390 1.00 KCNH2 (0.67) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL11914545 0.91 KCNH2 (0.79) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL378375 0.91 KCNH2 (0.79) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL11911820 0.91 KCNH2 (0.79) KCNH2DRD3DRD2CYP1A2CYP2D6
SCHEMBL378306 0.89 KCNH2 (0.68) KCNH2DRD3DRD2
Hydrochloric Acid SCHEMBL378883 0.88 KCNH2 (0.67) KCNH2DRD3DRD2
SCHEMBL11915309 0.86 KCNH2 (0.80) KCNH2DRD3DRD2CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745040-A1 AZABICYCLO(3.1.0) HEXANE DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2007-01-24 EP claimed
WO-2005080382-A1 AZABICYCLO (3.1.0) HEXANE DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2005-09-01 WO claimed