SCHEMBL5244069

SCHEMBL5244069

CCNC(=O)c1ccc(-n2cc(C(=O)NCCOc3ccccc3)nn2)c(OCCCCCCF)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.43
KMT2A Q03164 1/20 0.43
NPC1 O15118 7/20 0.42
RAB9A P51151 6/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
POLB P06746 2/20 0.41
HPGD P15428 1/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
RECQL P46063 1/20 0.41
TP53 P04637 1/20 0.40
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
SMPD1 P17405 1/20 0.39
CASP6 P55212 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246036 0.91 NPC1 (0.41) BRD4KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL5246108 0.90 BRD4 (0.47) BRD4NPC1RAB9ASMN1; SMN2POLB
SCHEMBL5245521 0.89 SMPD1 (0.41) BRD4KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL5247900 0.89 SMPD1 (0.44) BRD4TP53DRD2DRD4DRD3
SCHEMBL5244720 0.89 KMT2A (0.43) KMT2ANPC1RAB9ASMN1; SMN2HPGD
SCHEMBL5243860 0.89 SMPD1 (0.42) BRD4TP53SMPD1
SCHEMBL5244569 0.88 SMPD1 (0.41) BRD4KMT2ATP53SMPD1
SCHEMBL5247618 0.88 SMPD1 (0.43) BRD4POLBTP53DRD2DRD4
SCHEMBL5245878 0.88 BRD4 (0.42) BRD4KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL5244512 0.87 SMPD1 (0.42) BRD4KMT2APOLBTP53DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed