SCHEMBL5245285

SCHEMBL5245285

CCNC(=O)c1ccc(-n2cc(C(=O)NC3CCOCC3)nn2)c(OCCCCCCF)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.43
PLK1 P53350 2/20 0.40
PLK3 Q9H4B4 1/20 0.40
PLK2 Q9NYY3 1/20 0.40
ACKR3 P25106 1/20 0.39
WDR5 P61964 1/20 0.38
CNR2 P34972 6/20 0.38
FAAH O00519 2/20 0.37
F10 P00742 1/20 0.37
ACSS2 Q9NR19 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3112178 0.94 ACKR3 (0.41) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL3107180 0.94 ACKR3 (0.41) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL5246436 0.94 ACKR3 (0.44) PLK1PLK3PLK2ACKR3CNR2
SCHEMBL3110327 0.94 ACKR3 (0.42) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL5247636 0.91 ACKR3 (0.38) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL3110965 0.89 ACKR3 (0.43) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL5250118 0.88 BRD4 (0.43) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL3106830 0.87 MAPK14 (0.45) ACKR3CNR2
SCHEMBL3114010 0.87 CNR2 (0.40) BRD4PLK1PLK3PLK2ACKR3
SCHEMBL3113338 0.87 SMPD1 (0.43) BRD4PLK1PLK3PLK2ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed