SCHEMBL5252178

SCHEMBL5252178

O=C(Nc1cccc(Oc2ccc3cnn(C(c4cccs4)c4cccs4)c3c2)c1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.51
NR1H4 Q96RI1 1/20 0.46
HPSE Q9Y251 1/20 0.44
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
PLAU P00749 1/20 0.44
MAPT P10636 3/20 0.43
MAPK1 P28482 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
RECQL P46063 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
NLRP3 Q96P20 1/20 0.43
GALK1 P51570 1/20 0.43
CASP6 P55212 1/20 0.43
MCL1 Q07820 1/20 0.43
PLEC Q15149 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5252140 0.81 KDR (0.61) KDRNR1H4HPSEKCNK3KCNK9
SCHEMBL5249171 0.73 KDR (0.59) KDRNR1H4HPSEKCNK3KCNK9
SCHEMBL5250661 0.71 KDR (0.61) KDRNR1H4HPSEKCNK3KCNK9
SCHEMBL22543145 0.71 NR1H4 (0.78) NR1H4HPSEKCNK3KCNK9PLAU
SCHEMBL5253291 0.70 KDR (0.48) KDRNR1H4HPSEPLAUMAPT
SCHEMBL30396799 0.70 KCNK3 (0.71) KDRNR1H4HPSEKCNK3KCNK9
SCHEMBL6710523 0.69 KDR (0.51) KDRNR1H4HPSENPC1RAB9A
SCHEMBL5252137 0.68 KDR (1.00) KDRFGFR1
SCHEMBL20917283 0.67 CACNA2D1 (0.58) MAPTMAPK1MEN1KMT2ALMNA
SCHEMBL14684329 0.67 NR1H4 (0.71) NR1H4HPSEKCNK3KCNK9PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1614683-B1 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use AGOURON PHARMA (US) 2007-11-21 EP disclosed