SCHEMBL5253138

SCHEMBL5253138

COc1cc(-c2ccccc2C)ccc1C(=O)N1CCCC(CC(=O)N2CCN(C)CC2)c2cc(Cl)ccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 14/20 0.44
AVPR1A P37288 3/20 0.42
ABCB11 O95342 1/20 0.42
ADRB2 P07550 1/20 0.42
HTR1A P08908 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
CHRM1 P11229 1/20 0.42
TBXA2R P21731 1/20 0.42
HTR2C P28335 1/20 0.42
HRH1 P35367 1/20 0.42
OPRM1 P35372 1/20 0.42
GLP1R P43220 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
GPR119 Q8TDV5 1/20 0.42
HSD17B3 P37058 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9281226 0.93 AVPR2 (0.42) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL4687374 0.86 AVPR2 (0.60) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL7017339 0.85 AVPR2 (0.46) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL7017556 0.83 AVPR2 (0.46) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL4698258 0.82 AVPR2 (0.52) AVPR2AVPR1AABCB11ADRB2HTR1A
Hydrochloric Acid SCHEMBL7341607 0.81 AVPR2 (0.51) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL4682372 0.80 AVPR2 (0.50) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL7246942 0.80 AVPR2 (0.43) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL7334156 0.80 AVPR2 (0.51) AVPR2AVPR1AABCB11ADRB2HTR1A
SCHEMBL7022224 0.80 AVPR2 (0.38) AVPR2AVPR1AABCB11ADRB2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1221440-B1 Benzoheterocyclic derivatives useful as vasopressin or oxytocin modulators OTSUKA PHARMA CO LTD (JP) 2007-04-25 EP disclosed
EP-0765314-B1 BENZOHETEROCYCLIC DERIVATIVES USEFUL AS VASOPRESSIN OR OXYTOCIN MODULATORS OTSUKA PHARMA CO LTD (JP) 2003-05-07 EP disclosed
EP-1221440-A1 Benzoheterocyclic derivatives useful as vasopressin or oxytocin modulators Otsuka Pharmaceutical Company, Limited (JP) 2002-07-10 EP disclosed
EP-0765314-A1 BENZOHETEROCYCLIC DERIVATIVES USEFUL AS VASOPRESSIN OR OXYTOCIN MODULATORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-02 EP disclosed
WO-1995034540-A1 BENZOHETEROCYCLIC DERIVATIVES USEFUL AS VASOPRESSIN OR OXYTOCIN MODULATORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-12-21 WO disclosed