SCHEMBL5255341

SCHEMBL5255341

CC(C)(c1cc(-c2cccc(-c3cncc(C(O)(C(F)(F)F)C(F)(F)F)c3)c2)cc2cccnc12)S(C)(=O)=O

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 15/20 0.52
PDE4A P27815 6/20 0.42
PDE4B Q07343 6/20 0.42
PDE4C Q08493 6/20 0.42
PDE4D Q08499 6/20 0.42
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259329 0.91 CYP2C9 (0.56) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5255335 0.86 CYP2C9 (0.72) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5257729 0.83 CYP2C9 (0.69) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5262925 0.83 CYP2C9 (0.54) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5259631 0.82 CYP2C9 (0.58) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5260138 0.80 CYP2C9 (0.69) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5258285 0.78 CYP2C9 (0.52) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5261957 0.78 CYP2C9 (0.50) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5257780 0.78 CYP2C9 (0.50) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5255806 0.78 CYP2C9 (0.53) CYP2C9PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517895-B1 8-(BIARYL) QUINOLINE PDE4 INHIBITORS MERCK FROSST CANADA LTD (CA) 2007-03-14 EP claimed