SCHEMBL5255607

SCHEMBL5255607

CN1C(=O)C(c2cn(C)c3ccccc23)=C(c2cc(OCCN3CCOCC3)cc3ccoc23)C1=O

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 10/20 0.52
QPCT Q16769 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
EGFR P00533 1/20 0.41
CYP1A2 P05177 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4985394 0.92 GSK3B (0.53) GSK3BEGFRADORA3ADORA2AADORA2B
Hydrochloric Acid SCHEMBL5259095 0.90 GSK3B (0.63) GSK3BQPCT
SCHEMBL4991291 0.86 GSK3B (0.46) GSK3B
SCHEMBL4994634 0.86 GSK3B (0.46) GSK3B
SCHEMBL6581578 0.84 GSK3B (0.55) GSK3BQPCTNPC1RAB9AADORA2A
SCHEMBL4990655 0.83 GSK3B (0.44) GSK3B
SCHEMBL4985209 0.82 GSK3B (0.56) GSK3B
SCHEMBL4988608 0.76 CCNT1 (0.52) GSK3B
SCHEMBL6582702 0.76 GSK3B (0.56) GSK3BNPC1RAB9AADORA2AADORA1
SCHEMBL4987619 0.75 GSK3B (0.44) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487822-B1 PYRROLE-2,5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS LILLY CO ELI (US) 2007-08-01 EP disclosed