SCHEMBL5258367

SCHEMBL5258367

C[SiH](C)C(O)([C@@H]1CCC(=O)O1)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
CYP1A2 P05177 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9927430 0.77 CA1 (0.46) CA1CA9CYP1A2
SCHEMBL9607558 0.73 CA1 (0.50) CA1CA9CYP1A2
SCHEMBL2664154 0.73 CA1 (0.50) CA1CA9CYP1A2
SCHEMBL9607559 0.73 CA1 (0.50) CA1CA9CYP1A2
SCHEMBL9559189 0.73 CA1 (0.44) CA1CA9CYP1A2
SCHEMBL25327380 0.68 CA1 (0.41) CA1CA9CYP1A2
SCHEMBL3792494 0.67 CA1 (0.39) CA1CA9CYP1A2
SCHEMBL22972533 0.67 CA1 (0.43) CA1CA9CYP1A2
SCHEMBL27502798 0.67 CA1 (0.48) CA1CA9CYP1A2
SCHEMBL16449196 0.67 CA1 (0.36) CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242426-B1 GAMMA-HYDROXY-2-(FLUOROALKYLAMINOCARBONYL)-1-PIPERAZINEPENTANAMIDES AS HIV PROTEASE INHIBITORS MERCK & CO INC (US) 2007-10-31 EP disclosed
US-6642237-B1 Inhibitors of HIV protease and inhibitors of HIV replication, used in the prevention or treatment of infection by HIV and treatment for AIDS MERCK & CO., INC. 2003-11-04 US disclosed