SCHEMBL5260065

SCHEMBL5260065

Cc1c(N2CCC(C3(NC(=O)OC(C)(C)C)CC3)C2)cc(O)c2c(=O)c(C(=O)O)cn([C@@H]3C[C@H]3F)c12

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.47
KCNH2 Q12809 3/20 0.34
HRH3 Q9Y5N1 1/20 0.34
PIK3CD O00329 1/20 0.31
PIK3R1 P27986 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CG P48736 1/20 0.31
SCN5A Q14524 1/20 0.30
ALDH1A1 P00352 2/20 0.30
POLB P06746 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
TOP2A P11388 1/20 0.30
TOP2B Q02880 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2081948 1.00 CYP3A4 (0.47) CYP3A4KCNH2HRH3PIK3CDPIK3R1
SCHEMBL2081946 1.00 CYP3A4 (0.47) CYP3A4KCNH2HRH3PIK3CDPIK3R1
SCHEMBL2083026 0.83 CYP3A4 (0.63) CYP3A4KCNH2HRH3SCN5AALDH1A1
SCHEMBL2083029 0.83 CYP3A4 (0.63) CYP3A4KCNH2HRH3SCN5AALDH1A1
SCHEMBL2081994 0.82 CYP3A4 (0.58) CYP3A4KCNH2PIK3CGALDH1A1POLB
SCHEMBL2081996 0.82 CYP3A4 (0.58) CYP3A4KCNH2PIK3CGALDH1A1POLB
SCHEMBL482753 0.81 CYP3A4 (0.72) CYP3A4KCNH2ALDH1A1POLBOPRM1
SCHEMBL2080690 0.80 CYP3A4 (0.51) CYP3A4KCNH2HRH3SCN5AALDH1A1
SCHEMBL2080688 0.80 CYP3A4 (0.51) CYP3A4KCNH2HRH3SCN5AALDH1A1
SCHEMBL14014253 0.79 CYP3A4 (0.45) CYP3A4KCNH2ALDH1A1POLBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1336611-B1 DEHALOGENO COMPOUNDS DAIICHI SEIYAKU CO (JP) 2007-09-05 EP disclosed