SCHEMBL5260615

SCHEMBL5260615

CC(C)(c1cc(-c2cccc(-c3cccs3)c2)cc2cccnc12)S(C)(=O)=O

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 14/20 0.53
PDE4A P27815 6/20 0.44
PDE4B Q07343 6/20 0.44
PDE4C Q08493 6/20 0.44
PDE4D Q08499 6/20 0.44
GLO1 Q04760 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5260138 0.86 CYP2C9 (0.69) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5261474 0.84 CYP2C9 (0.48) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5259110 0.83 CYP2C9 (0.69) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5257729 0.83 CYP2C9 (0.69) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5262232 0.83 CYP2C9 (0.57) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5258650 0.82 CYP2C9 (0.70) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5257427 0.82 CYP2C9 (0.75) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5262206 0.81 CYP2C9 (0.55) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5258956 0.81 CYP2C9 (0.51) CYP2C9PDE4APDE4BPDE4CPDE4D
SCHEMBL5257886 0.81 CYP2C9 (0.51) CYP2C9PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517895-B1 8-(BIARYL) QUINOLINE PDE4 INHIBITORS MERCK FROSST CANADA LTD (CA) 2007-03-14 EP claimed