SCHEMBL5264183

SCHEMBL5264183

CCn1c(=O)c2c(ncn2CCCCO)n(CC)c1=O

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.67
PDE4B Q07343 7/20 0.67
PDE4C Q08493 7/20 0.67
PDE4D Q08499 7/20 0.67
ADORA2A P29274 5/20 0.56
ADORA2B P29275 5/20 0.53
CNOT7 Q9UIV1 5/20 0.52
LMNA P02545 2/20 0.51
ESR1 P03372 1/20 0.49
CYP1A2 P05177 1/20 0.49
MAPT P10636 1/20 0.49
NFKB1 P19838 1/20 0.49
ACHE P22303 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9294207 0.99 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL5239597 0.96 PDE4A (0.72) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL5235343 0.90 PDE4A (0.71) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9294503 0.90 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9294305 0.90 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL8362364 0.86 RXFP1 (0.67) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10761423 0.85 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10811726 0.84 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL10815947 0.84 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL8912388 0.84 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1829523-A1 Cosmetic use of an N-oxide derivative of theophylline L'OREAL (FR) 2007-09-05 EP disclosed