SCHEMBL5264483

SCHEMBL5264483

ClCc1ccc(OCCNC2CCCCC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.66
CYP1A2 P05177 1/20 0.66
CYP2D6 P10635 1/20 0.66
CYP2C19 P33261 1/20 0.66
ALDH1A1 P00352 7/20 0.61
FOXM1 Q08050 2/20 0.61
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.53
HPGD P15428 1/20 0.52
HRH3 Q9Y5N1 1/20 0.51
TDP1 Q9NUW8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1984254 0.98 KDM4E (0.64) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
Hydrochloric Acid SCHEMBL1988261 0.97 KDM4E (0.66) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL7140903 0.82 KDM4E (0.79) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL23074654 0.81 KDM4E (0.88) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL23074658 0.81 KDM4E (0.88) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL2352175 0.81 KDM4E (0.69) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL7135308 0.81 KDM4E (0.81) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL12204238 0.80 KDM4E (0.70) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL11876550 0.78 KDM4E (0.58) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL1299936 0.78 KDM4E (0.64) KDM4ECYP1A2CYP2D6CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1796664-A1 NOVEL TETRACYCLIC HETEROATOM CONTAINING DERIVATIVES USEFUL AS SEX STEROID HORMONE RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2007-06-20 EP disclosed
WO-2006047017-A1 NOVEL TETRACYCLIC HETEROATOM CONTAINING DERIVATIVES USEFUL AS SEX STEROID HORMONE RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-04 WO disclosed