SCHEMBL5266299

SCHEMBL5266299

Cc1[nH]c(C(=O)Nc2ccc(-c3cnc(Cl)c(C(=O)O)c3C)cc2)c(Cl)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
PIK3C3 Q8NEB9 2/20 0.43
DAO P14920 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4901768 0.80 DAO (0.46) DAO
SCHEMBL5266303 0.77 DAO (0.45) DAO
SCHEMBL4910360 0.75 PTPN1 (0.49)
SCHEMBL29717252 0.75 TOP2A (0.56) NPC1PKMRAB9ADAO
SCHEMBL4903739 0.74 SCN10A (0.51) DAO
SCHEMBL4907263 0.74 IKBKE (0.44) DAO
SCHEMBL5256434 0.73 NPC1 (0.42) NPC1PKMRAB9ADAO
SCHEMBL4909723 0.73 TOP2A (0.49)
SCHEMBL4907614 0.72 TOP2A (0.42) DAO
SCHEMBL5263131 0.72 HPGD (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861393-A2 PYRROLE DERIVATIVES AS DNA GYRASE AND TOPOISOMERASE INHIBITORS AstraZeneca AB (SE) 2007-12-05 EP claimed
WO-2006092599-A2 PYRROLE DERIVATIVES AS DNA GYRASE AND TOPOISOMERASE INHIBITORS ASTRAZENECA AB (SE) 2006-09-08 WO claimed