SCHEMBL5266537

SCHEMBL5266537

O=c1c(Br)c(OCCc2ccccc2)ncn1Cc1cccc(F)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.52
KDM4E B2RXH2 2/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAPT P10636 6/20 0.43
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
PDE1C Q14123 2/20 0.41
PDE1A P54750 1/20 0.41
PDE1B Q01064 1/20 0.41
LMNA P02545 3/20 0.41
THRB P10828 1/20 0.40
MMP13 P45452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3519707 0.89 MAPK14 (0.59) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3521113 0.86 MAPK14 (0.58) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3521534 0.85 MAPK14 (0.67) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3526494 0.83 MAPK14 (0.49) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3521221 0.81 MAPK14 (0.48) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3520032 0.81 MAPK14 (0.51) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3521293 0.81 MAPK14 (0.46) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3519362 0.81 MAPK14 (0.51) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3520704 0.81 MAPK14 (0.53) MAPK14KDM4EHPGDNPSR1MAPT
SCHEMBL3518775 0.81 MAPK14 (0.69) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753731-A2 PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE AS P38 KINASE MODULATORS Pharmacia Corporation (US) 2007-02-21 EP disclosed
WO-2004087677-A2 PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE AS P38 KINASE MODULATORS PHARMACIA CORPORATION (US) 2004-10-14 WO disclosed