SCHEMBL5267732

SCHEMBL5267732

Cc1cccnc1COc1ncc(C(=O)NC2CCCC[C@H]2O)cc1-c1ccc(F)cc1

nearest known ligand 0.69

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 0.69
TACR2 P21452 1/20 0.58
CNR2 P34972 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1380828 1.00 CNR1 (0.69) CNR1TACR2CNR2
SCHEMBL3846966 0.92 CNR1 (0.79) CNR1TACR2CNR2
SCHEMBL3845283 0.86 CNR1 (0.84) CNR1TACR2CNR2
SCHEMBL5918463 0.86 CNR1 (0.84) CNR1TACR2CNR2
SCHEMBL3848299 0.86 CNR1 (0.84) CNR1TACR2CNR2
SCHEMBL1381869 0.84 CNR1 (0.84) CNR1TACR2CNR2
SCHEMBL5348881 0.84 CNR1 (0.84) CNR1TACR2CNR2
SCHEMBL3848484 0.83 CNR1 (0.71) CNR1TACR2CNR2
SCHEMBL1376863 0.83 CNR1 (0.83) CNR1TACR2CNR2
SCHEMBL2703819 0.82 CNR1 (0.77) CNR1TACR2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1868999-A1 PYRIDINE-3-CARBOXAMIDE DERIVATIVES AS CB1 INVERSE AGONISTS F. Hoffmann-Roche AG (CH) 2007-12-26 EP disclosed
WO-2006106054-A1 PYRIDINE-3-CARBOXAMIDE DERIVATIVES AS CB1 INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-10-12 WO disclosed