SCHEMBL5281609

SCHEMBL5281609

COc1ccc(-c2ccncc2O[C@H]2SC[C@@H](OC(C)=O)[C@H](OC(C)=O)[C@H]2OC(C)=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.39
CACNA1B Q00975 1/20 0.38
BACE1 P56817 1/20 0.37
RPS6KA3 P51812 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
SYK P43405 2/20 0.35
AURKB Q96GD4 1/20 0.35
INCENP Q9NQS7 1/20 0.35
GABRA1 P14867 4/20 0.34
GABRB2 P47870 2/20 0.34
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA3 P34903 2/20 0.33
GABRA2 P47869 2/20 0.33
STIM1 Q13586 1/20 0.33
ORAI1 Q96D31 1/20 0.33
GABRA5 P31644 1/20 0.33
CYP2D6 P10635 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2139628 1.00 SLC22A12 (0.39) SLC22A12CACNA1BBACE1RPS6KA3GSK3A
SCHEMBL314690 0.91 SLC22A12 (0.32) SLC22A12
SCHEMBL314689 0.91 SLC22A12 (0.32) SLC22A12
SCHEMBL2141893 0.89 CACNA1B (0.38) SLC22A12CACNA1BRPS6KA3GSK3AGSK3B
SCHEMBL2141887 0.89 CACNA1B (0.38) SLC22A12CACNA1BRPS6KA3GSK3AGSK3B
SCHEMBL316662 0.87 MKNK1 (0.36) SLC22A12ALDH1A1CYP2C9CYP2C19
SCHEMBL316661 0.87 MKNK1 (0.36) SLC22A12ALDH1A1CYP2C9CYP2C19
SCHEMBL2142874 0.86 SLC22A12 (0.41) SLC22A12GSK3AGSK3BAURKB
SCHEMBL2141335 0.86 CACNA1B (0.40) SLC22A12CACNA1BBACE1
SCHEMBL2141327 0.86 CACNA1B (0.40) SLC22A12CACNA1BBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861411-A2 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF LABORATOIRES FOURNIER S.A. (FR) 2007-12-05 EP disclosed
WO-2006100413-A9 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF FOURNIER LAB SA (FR) 2007-10-18 WO disclosed
WO-2006100413-A2 NOVEL COMPOUNDS DERIVED FROM 5-THIOXYLOSE AND THERAPEUTIC USE THEREOF LABORATOIRES FOURNIER S.A. (FR) 2006-09-28 WO disclosed