SCHEMBL5283535

SCHEMBL5283535

CC(C)(C)OC(=O)N1CCN(Cc2ccc(I)cc2)C(=O)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.49
DPP4 P27487 3/20 0.48
HDAC1 Q13547 4/20 0.46
HDAC6 Q9UBN7 4/20 0.46
VEGFA P15692 1/20 0.43
EGLN1 Q9GZT9 1/20 0.43
NR1H2 P55055 2/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ESR2 Q92731 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
STS P08842 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
PREP P48147 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20129614 0.89 TP53 (0.50) TP53DPP4HDAC1HDAC6VEGFA
SCHEMBL22532823 0.89 TP53 (0.50) TP53DPP4HDAC1HDAC6VEGFA
SCHEMBL14103789 0.89 VEGFA (0.53) TP53HDAC1HDAC6VEGFAEGLN1
SCHEMBL1876106 0.88 TP53 (0.49) TP53HDAC1HDAC6VEGFAEGLN1
SCHEMBL4297578 0.88 NR1H2 (0.50) TP53DPP4HDAC1HDAC6VEGFA
SCHEMBL4158417 0.88 DPP4 (0.49) TP53DPP4HDAC1HDAC6VEGFA
SCHEMBL1049753 0.88 HDAC1 (0.50) TP53DPP4HDAC1HDAC6KMT2A
SCHEMBL1081669 0.87 HDAC1 (0.50) TP53HDAC1HDAC6VEGFAEGLN1
SCHEMBL2262766 0.87 CYP3A4 (0.52) TP53DPP4HDAC1HDAC6SMN1; SMN2
SCHEMBL5328156 0.86 TP53 (0.47) TP53DPP4HDAC1HDAC6VEGFA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007008144-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES AS INHIBITORS OF FACTOR XA ASTRAZENECA AB (SE) 2007-01-18 WO disclosed