SCHEMBL529400

SCHEMBL529400

CN(C(=O)O)C1CCCN(c2ccc([N+](=O)[O-])cn2)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.56
ALDH1A1 P00352 6/20 0.55
LMNA P02545 3/20 0.55
ALOX12 P18054 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
L3MBTL1 Q9Y468 2/20 0.53
POLB P06746 1/20 0.53
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
ATM Q13315 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
HPGD P15428 1/20 0.47
NPY2R P49146 1/20 0.47
MAPK1 P28482 2/20 0.44
PKM P14618 1/20 0.44
NPBWR1 P48145 1/20 0.43
MCHR1 Q99705 1/20 0.43
KDM4E B2RXH2 1/20 0.42
PANK3 Q9H999 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529399 1.00 MAPT (0.56) MAPTALDH1A1LMNAALOX12NPSR1
SCHEMBL528903 0.93 MAPT (0.59) MAPTALDH1A1LMNAALOX12NPSR1
SCHEMBL528904 0.93 MAPT (0.59) MAPTALDH1A1LMNAALOX12NPSR1
SCHEMBL15191254 0.86 RET (0.51) MAPTALDH1A1LMNAALOX12NPSR1
SCHEMBL529250 0.82 BTK (0.48) MAPTALDH1A1NPSR1KMT2AHPGD
SCHEMBL24267753 0.80 MAPT (0.66) MAPTALDH1A1LMNAALOX12NPSR1
SCHEMBL595593 0.79 MAPT (0.53) MAPTALDH1A1LMNAALOX12NPSR1
SCHEMBL23089642 0.79 MAPT (0.56) MAPTALDH1A1POLBMEN1KMT2A
SCHEMBL23089638 0.79 MAPT (0.56) MAPTALDH1A1POLBMEN1KMT2A
SCHEMBL2792238 0.79 MAPT (0.68) MAPTALDH1A1LMNAALOX12NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed