SCHEMBL529464

SCHEMBL529464

CC(C)C(=O)c1cnc2ccc(-c3ccc(C#N)nc3)cc2c1NC1CCCCC1NC(=O)O

nearest known ligand 0.71

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MELK Q14680 15/20 0.71
TNF P01375 1/20 0.44
ATM Q13315 3/20 0.42
ATR Q13535 2/20 0.42
KCNH2 Q12809 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15191360 0.89 MELK (0.82) MELKIRAK4
SCHEMBL15191359 0.89 MELK (0.82) MELKIRAK4
SCHEMBL15197597 0.83 MELK (0.85) MELKIRAK4
SCHEMBL15191641 0.83 MELK (1.00) MELK
SCHEMBL15191643 0.83 MELK (1.00) MELK
SCHEMBL529166 0.83 MELK (0.70) MELK
SCHEMBL530025 0.83 MELK (0.70) MELK
SCHEMBL529512 0.81 MELK (0.73) MELKTNFATMATRKCNH2
SCHEMBL529607 0.81 MELK (0.46) MELKATMATRKCNH2
SCHEMBL15191202 0.80 MELK (0.75) MELKIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed