SCHEMBL5306457

SCHEMBL5306457

Clc1ccc(Cn2cncn2)cc1Cl

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.61
KMT2A Q03164 2/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
CCR1 P32246 1/20 0.47
CCR2 P41597 1/20 0.47
CCR4 P51679 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17159812 0.85 CYP19A1 (0.80) CYP19A1HDAC1HDAC6
SCHEMBL11354103 0.82 CYP19A1 (0.69) CYP19A1KMT2AMEN1ALDH1A1HDAC1
Hydrochloric Acid SCHEMBL11358575 0.80 CYP19A1 (0.67) CYP19A1KMT2AMEN1ALDH1A1HDAC1
SCHEMBL15688800 0.80 CYP19A1 (0.71) CYP19A1HDAC1HDAC6
SCHEMBL9525426 0.79 KDM4E (0.50) CYP19A1ALDH1A1HDAC1HDAC6
SCHEMBL3235365 0.78 CYP19A1 (0.69) CYP19A1HDAC1HDAC6
SCHEMBL31415788 0.77 HRH4 (0.45) CYP19A1KMT2ATSHRMAPK1HSD17B10
Hydrochloric Acid SCHEMBL11347612 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1HDAC1HDAC6
SCHEMBL306232 0.77 CYP19A1 (0.67) CYP19A1HDAC1HDAC6
SCHEMBL307542 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007014054-A2 BENZENESULFONAMIDE INHIBITOR OF CCR2 CHEMOKINE RECEPTOR GLAXO GROUP LIMTED (GB) 2007-02-01 WO disclosed
WO-2007014054-A2 BENZENESULFONAMIDE INHIBITOR OF CCR2 CHEMOKINE RECEPTOR GLAXO GROUP LIMTED (GB) 2007-02-01 WO disclosed