SCHEMBL5307889

SCHEMBL5307889

Cc1nc(NC(=O)CCNCCN2CCOCC2)sc1-c1ccnc(Nc2ccc(Cl)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.48
CLK1 P49759 2/20 0.48
NPC1 O15118 1/20 0.48
TSHR P16473 1/20 0.48
RAB9A P51151 1/20 0.48
KMT2A Q03164 8/20 0.46
MEN1 O00255 7/20 0.46
MAPT P10636 6/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
ALOX12 P18054 2/20 0.46
GAA P10253 2/20 0.46
TNIK Q9UKE5 1/20 0.45
HPGD P15428 3/20 0.44
PIK3CG P48736 3/20 0.44
KDM4E B2RXH2 2/20 0.44
NPSR1 Q6W5P4 2/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704253 0.86 CDK2 (0.53) ALDH1A1CLK1KMT2AMEN1MAPT
SCHEMBL12841836 0.80 CDK2 (0.55) ALDH1A1CLK1NPC1TSHRRAB9A
SCHEMBL2073904 0.79 CDK2 (0.57) ALDH1A1CLK1KMT2AMEN1MAPT
SCHEMBL5245918 0.75 GAA (0.46) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E
SCHEMBL27624139 0.75 CDK2 (0.52) ALDH1A1CLK1NPC1TSHRRAB9A
SCHEMBL2074524 0.71 CDK2 (0.57) CLK1TNIK
SCHEMBL2075857 0.70 CDK2 (0.56) CLK1GAATNIK
SCHEMBL2075970 0.69 MEN1 (0.53) ALDH1A1KMT2AMEN1MAPTSMN1; SMN2
SCHEMBL14851611 0.67 PIK3CG (0.72) ALDH1A1CLK1NPC1TSHRRAB9A
SCHEMBL924953 0.67 PIK3CA (0.56) ALDH1A1CLK1NPC1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1864983-A1 PYRIMIDINE COMPOUNDS AS CYCLIN-DEPENDENT KINASE INHIBITORS Cyclacel Limited (GB) 2007-12-12 EP claimed