SCHEMBL5308270

SCHEMBL5308270

O=C(O)CNC(=O)c1c(O)c2ccccc2n(CCC2CC2)c1=O

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.74
EGLN1 Q9GZT9 2/20 0.67
BBOX1 O75936 1/20 0.66
ASPH Q12797 1/20 0.66
KDM8 Q8N371 1/20 0.66
MEN1 O00255 8/20 0.55
KMT2A Q03164 8/20 0.55
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 1/20 0.55
HPGD P15428 1/20 0.55
HTT P42858 1/20 0.55
POLB P06746 1/20 0.55
GAA P10253 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
LMNA P02545 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8237984 0.95 HIF1A (0.68) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL8243641 0.85 HIF1A (0.67) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL17578541 0.85 HIF1A (1.00) HIF1A
SCHEMBL8244798 0.84 HIF1A (0.67) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL2085626 0.83 HIF1A (0.59) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL2382364 0.83 EGLN1 (0.78) EGLN1MEN1KMT2AKDM4EALDH1A1
SCHEMBL8244110 0.82 EGLN1 (0.70) EGLN1MEN1KMT2AKDM4EALDH1A1
SCHEMBL8247183 0.82 HIF1A (0.62) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL8244097 0.81 EGLN1 (0.69) EGLN1MEN1KMT2AKDM4EALDH1A1
SCHEMBL5310453 0.81 EGLN1 (0.69) EGLN1MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007038571-A2 PROLYL HYDROXYLASE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-05 WO claimed
WO-2007038571-A2 PROLYL HYDROXYLASE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-05 WO disclosed