SCHEMBL5314059

SCHEMBL5314059

CN(C)Cc1ccc(N/C(=C2/C(=O)Nc3cc(F)ccc32)c2ccc(CCC(=O)O)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.41
MCHR1 Q99705 3/20 0.38
NR1H4 Q96RI1 1/20 0.38
FFAR1 O14842 8/20 0.37
FFAR4 Q5NUL3 5/20 0.36
PPARG P37231 1/20 0.36
AURKA O14965 1/20 0.35
TGM2 P21980 1/20 0.35
LIMK2 P53671 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
NCOR2 Q9Y618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL228447 1.00 BACE1 (0.41) BACE1MCHR1NR1H4FFAR1FFAR4
SCHEMBL228448 1.00 BACE1 (0.41) BACE1MCHR1NR1H4FFAR1FFAR4
Hydrochloric Acid SCHEMBL1943757 0.99 BACE1 (0.41) BACE1MCHR1NR1H4FFAR1FFAR4
Hydrochloric Acid SCHEMBL1943759 0.99 BACE1 (0.41) BACE1MCHR1NR1H4FFAR1FFAR4
SCHEMBL224596 0.93 BACE1 (0.41) BACE1NR1H4FFAR1FFAR4PPARG
SCHEMBL224595 0.93 BACE1 (0.41) BACE1NR1H4FFAR1FFAR4PPARG
SCHEMBL228645 0.92 BACE1 (0.38) BACE1NR1H4FFAR1FFAR4PPARG
SCHEMBL228644 0.92 BACE1 (0.38) BACE1NR1H4FFAR1FFAR4PPARG
SCHEMBL225215 0.92 BACE1 (0.39) BACE1NR1H4FFAR1FFAR4PPARG
SCHEMBL225379 0.92 BACE1 (0.43) BACE1FFAR1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007057399-A2 TREATMENT OF CANCER WITH INDOLE DERIVATIVES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-24 WO disclosed