SCHEMBL5315670

SCHEMBL5315670

Oc1c(F)cc(F)cc1[AsH2]

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.46
CA9 Q16790 2/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
IDO1 P14902 1/20 0.38
NOTUM Q6P988 1/20 0.37
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CES2 O00748 3/20 0.35
CES1 P23141 3/20 0.35
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
TTR P02766 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78286 0.80 ERN1 (0.56) ERN1CA9CA12CA1IDO1
SCHEMBL27540052 0.77 ERN1 (0.54) ERN1CA9CA12CA1IDO1
SCHEMBL5310503 0.75 IDO1 (0.43) CA9CA12CA1IDO1PTGS1
SCHEMBL5513552 0.75 ERN1 (0.52) ERN1CA9CA12CA1IDO1
SCHEMBL8059874 0.72 IDO1 (0.55) ERN1CA9CA12CA1IDO1
SCHEMBL5399616 0.68 ERN1 (0.46) ERN1CA9CA12CA1IDO1
SCHEMBL1521925 0.68 ERN1 (0.46) ERN1CA9CA12CA1IDO1
SCHEMBL1155741 0.68 ERN1 (0.46) ERN1CA9CA12CA1IDO1
SCHEMBL12023112 0.68 PTGS1 (0.50) ERN1CA9CA12CA1IDO1
SCHEMBL104581 0.68 ERN1 (0.46) ERN1CA9CA12CA1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765795-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Addex Pharmaceuticals SA (CH) 2007-03-28 EP disclosed
WO-2005123703-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMACEUTICALS SA (CH) 2005-12-29 WO disclosed