SCHEMBL5318949

SCHEMBL5318949

C[S+]([O-])c1ccc(/C(=C/c2cccc(-c3cc(C(C)(C)S(C)(=O)=O)cc4cccnc34)c2)c2ccc(C(C)(C)O)cn2)cc1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 13/20 0.59
PDE4B Q07343 13/20 0.59
PDE4C Q08493 13/20 0.59
PDE4D Q08499 13/20 0.59
CYP2C9 P11712 9/20 0.59
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7088307 0.92 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027178 0.92 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027181 0.92 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027184 0.92 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DCYP2C9
Quinoline SCHEMBL27575381 0.88 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4034289 0.84 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4034297 0.84 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4034294 0.84 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL7449314 0.78 PDE4A (0.73) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL6988514 0.78 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633306-A4 USE OF PHOSPHATASE INHIBITORS AS ADJUNCT THERAPY FOR PSYCHIATRIC DISORDERS MERCK & CO INC (US) 2007-05-16 EP disclosed
EP-1633306-A2 USE OF PHOSPHATASE INHIBITORS AS ADJUNCT THERAPY FOR PSYCHIATRIC DISORDERS Merck & Co., Inc. (US) 2006-03-15 EP disclosed
WO-2004105698-A2 USE OF PHOSPHATASE INHIBITORS AS ADJUNCT THERAPY FOR PSYCHIATRIC DISORDERS MERCK & CO., INC. (US) 2004-12-09 WO disclosed