SCHEMBL5319277

SCHEMBL5319277

Cc1ccc(-c2nc(N)nc(O)c2C#N)cc1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 16/20 0.70
ADORA2A P29274 14/20 0.70
ADORA2B P29275 3/20 0.50
KMT2A Q03164 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321086 0.81 ADORA1 (0.70) ADORA1ADORA2AADORA2BKMT2ACYP1A2
SCHEMBL27573259 0.79 ADORA1 (0.67) ADORA1ADORA2AADORA2BKMT2ACYP1A2
SCHEMBL4904033 0.74 ADORA1 (0.77) ADORA1ADORA2AADORA2BKMT2AMEN1
SCHEMBL11175169 0.73 ADORA1 (0.45) ADORA1ADORA2AADORA2BKMT2ACYP1A2
SCHEMBL13045873 0.72 ADORA1 (0.57) ADORA1ADORA2AADORA2BKMT2ACYP1A2
SCHEMBL5321147 0.71 ADORA1 (0.77) ADORA1ADORA2AADORA2B
SCHEMBL4899129 0.71 ADORA1 (0.53) ADORA1ADORA2AADORA2BKMT2ACYP1A2
SCHEMBL6440910 0.71 ADORA1 (1.00) ADORA1ADORA2AADORA2B
SCHEMBL18356737 0.70 ADORA1 (0.71) ADORA1ADORA2AKMT2AMEN1ALDH1A1
SCHEMBL8914694 0.69 ADORA1 (0.54) ADORA1ADORA2AADORA2BKMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007098835-A1 AMINO PYRYMIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-09-07 WO disclosed
WO-2007098835-A1 AMINO PYRYMIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-09-07 WO disclosed