SCHEMBL532003

SCHEMBL532003

CCNC(=O)c1ccc(N2CCN(Cc3cc4c(c(OC)c3)OCON4)CC2)c(C)c1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.69
TNK2 Q07912 1/20 0.47
TNK1 Q13470 1/20 0.47
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532272 0.86 PARP1 (0.75) PARP1TNK2TNK1DRD2
SCHEMBL531932 0.82 PARP1 (1.00) PARP1
SCHEMBL532169 0.78 PARP1 (0.64) PARP1TNK1
SCHEMBL532488 0.78 PARP1 (0.75) PARP1DRD2DRD3
SCHEMBL532132 0.76 PARP1 (0.77) PARP1TNK2TNK1
SCHEMBL532023 0.75 PARP1 (1.00) PARP1
SCHEMBL532342 0.74 PARP1 (0.86) PARP1
SCHEMBL531939 0.74 PARP1 (1.00) PARP1
SCHEMBL532968 0.74 PARP1 (1.00) PARP1
SCHEMBL532080 0.73 PARP1 (0.84) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415767-A1 Poly (ADP-ribose) Polymerase (PARP) Inhibitors Takeda Pharmaceutical Company Limited (JP) 2012-02-08 EP disclosed