SCHEMBL5320194

SCHEMBL5320194

Nc1ncc(-c2ccc(F)cc2)nc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 3/20 0.48
NOS1 P29475 1/20 0.46
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 3/20 0.45
KDM4E B2RXH2 3/20 0.45
HPGD P15428 3/20 0.45
CYP3A4 P08684 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
ALDH1A1 P00352 3/20 0.44
ALOX5 P09917 1/20 0.44
RAB9A P51151 1/20 0.44
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
CYP2C9 P11712 2/20 0.41
ADORA1 P30542 3/20 0.39
ADORA2A P29274 2/20 0.39
PTK2B Q14289 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321269 0.82 NPC1 (0.50) ATRCYP1A2CYP2C19KDM4ECYP3A4
SCHEMBL23064174 0.82 PIK3CG (0.54) ATRHPGDMAPK1ALDH1A1
SCHEMBL12198422 0.82 ATR (0.48) ATRNOS1CYP2C19KDM4EHPGD
SCHEMBL31638393 0.81 ATR (0.51) ATRNOS1KDM4EL3MBTL1MAPK1
SCHEMBL934804 0.81 ATR (0.51) ATRNOS1KDM4EL3MBTL1MAPK1
SCHEMBL5318316 0.79 ATR (0.48) ATRNOS1CYP1A2CYP2C19KDM4E
SCHEMBL27983733 0.79 ATR (0.36) ATRALOX5APFEN1ADORA1ADORA2A
SCHEMBL934180 0.78 ATR (0.51) ATRNOS1KDM4EHPGDMAPK1
SCHEMBL20839008 0.78 ALOX5AP (0.39) ATRCYP3A4HTTALOX5APFEN1
SCHEMBL29911247 0.78 ALOX5AP (0.39) ATRCYP3A4HTTALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed