SCHEMBL5323846

SCHEMBL5323846

CC1(C(=O)O)CC(O)CN1S(=O)(=O)c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ALDH1A1 P00352 2/20 0.46
MMP2 P08253 1/20 0.42
CHRM1 P11229 1/20 0.41
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
CTSG P08311 1/20 0.39
CMA1 P23946 1/20 0.39
AKR1C3 P42330 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
GPR183 P32249 1/20 0.38
GRIN2B Q13224 2/20 0.37
RORC P51449 1/20 0.37
AKR1C1 Q04828 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201573 1.00 MEN1 (0.49) MEN1KMT2AALDH1A1MMP2CHRM1
SCHEMBL6296895 1.00 MEN1 (0.49) MEN1KMT2AALDH1A1MMP2CHRM1
SCHEMBL6296896 1.00 MEN1 (0.49) MEN1KMT2AALDH1A1MMP2CHRM1
SCHEMBL5201579 1.00 MEN1 (0.49) MEN1KMT2AALDH1A1MMP2CHRM1
SCHEMBL5200881 0.88 CNR1 (0.41) MEN1KMT2AAKR1C3
SCHEMBL5201586 0.88 CNR1 (0.41) MEN1KMT2AAKR1C3
SCHEMBL5201582 0.88 CNR1 (0.41) MEN1KMT2AAKR1C3
SCHEMBL5200884 0.88 CNR1 (0.41) MEN1KMT2AAKR1C3
SCHEMBL5201963 0.87 MEN1 (0.40) MEN1KMT2AALDH1A1MMP2CHRM1
SCHEMBL5201960 0.87 MEN1 (0.40) MEN1KMT2AALDH1A1MMP2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389200-A4 SUBSTITUTED N-ARYLSULFONYL-PROLINE DERIVATIVES AS POTENT CELL ADHESION INHIBITORS MERCK & CO INC (US) 2007-03-28 EP disclosed
EP-1389200-A1 SUBSTITUTED N-ARYLSULFONYL-PROLINE DERIVATIVES AS POTENT CELL ADHESION INHIBITORS Merck & Co., Inc. (US) 2004-02-18 EP disclosed
WO-2002074761-A1 SUBSTITUTED N-ARYLSULFONYL-PROLINE DERIVATIVES AS POTENT CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 2002-09-26 WO disclosed